2020
1) Discovery of a Novel Unsymmetrical Structural Class of HCV NS5A Inhibitors with Low Picomolar Antiviral Activity
H. Nakamura, Y. Akagi, T. Terui, S. Fujioka, Y. Komoda, W. Kinoshita, K. Maeda, Y. Ukaji, T. Inaba
Bioorg. Med. Chem. Lett. 2020, 30, 126932. DOI:org/10.1016/j.bmcl.2019.126932
2) 多点認識型含窒素複素環カルベンの開発と触媒的不斉反応への展開
Development of multi-functional NHC catalysts bearing pyridine moiety: Application to catalytic asymmetric reactions
T. Soeta, Y. Ukaji
有機合成化学協会誌; J. Synth. Org. Chem. Jpn. 2020, 78, 338−349. DOI:org/10.1016/j.bmcl.2019.126932
3) Orally Bioavailable HCV NS5A Inhibitors of Unsymmetrical Structural Class
H. Nakamura, S. Fujioka, T. Terui, S. Okuda, K. Kondo, Y. Tamatani, Y. Akagi, Y. Komoda, W. Kinoshita, S. Ito, K. Maeda, Y. Ukaji, T. Inaba
Bioorg. Med. Chem. Lett. 2020, 30, 127361. DOI.org/10.1016/j.bmcl.2020.127361
4) Synthesis of 3,6-Dihydro-2H-1,2-oxazines via Dimethylsulfoxonium Methylide Addition to α,β-Unsaturated Nitrones
M. Hasegawa, T. Suga, T. Soeta, Y. Ukaji
J. Org. Chem. 2020, 85, 11258−11264. doi.org/10.1021/acs.joc.0c01349
5) One-Shot Radical Cross Coupling Between Benzyl Alcohols and Alkenyl Halides using Ni/Ti/Mn System
T. Suga, Y. Takahashi, Y. Ukaji
Adv. Synth. Catal. 2020, 362, 5622-5626. doi.org/10.1002/adsc.202000945
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